Seletracetam (ucb 44212) inhibits high-voltage-activated Ca2+ currents and intracellular Ca2+ increase in rat cortical neurons in vitro
Articolo
Data di Pubblicazione:
2009
Abstract:
We analyzed the effects of seletracetam (ucb 44212; SEL), a new antiepileptic drug candidate, in an in vitro model of epileptic activity. The activity of SEL was compared to the effects of levetiracetam (LEV; Keppra), in the same assays.
Tipologia CRIS:
1.1 Articolo in rivista
Keywords:
Animals; Calcium; Dose-Response Relationship; Drug; Pyrrolidinones; Bicuculline; Calcium Channel Blockers; Neural Inhibition; Biophysics; Rats; Calcium Channels; GABA Antagonists; Patch-Clamp Techniques; Neurons; Rats; Wistar; Potassium Channel Blockers; Piracetam; Membrane Potentials; 4-Aminopyridine; Magnesium; Neocortex; Anticonvulsants; Male
Elenco autori:
Martella, Giuseppina; Bonsi, P; Sciamanna, Giuseppe; Platania, P; Madeo, Graziella; Tassone, A; Cuomo, D; Pisani, Antonio
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