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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Rivista
Codice:
E060692
ISSN:
0223-5234
Dati Generali
Dati Generali
Pubblicazioni (54)
Pulisci
Ordina Pubblicazioni:
ascendente
decrescente
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity
Articolo
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation.
Articolo
Advancing the antituberculosis activity of nitropicolinic acids and amides
Articolo
An efficient steroid pharmacophore-based strategy to identify new aromatase inhibitors
Articolo
Anti-tumor-promoting activity of simple models of galactoglycerolipids with branched and unsaturated acyl chains
Articolo
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections
Articolo
Benzothiozinone derivatives with anti-tubercular Activity−Further side chain investigation
Articolo
Bioisosteric replacement based on 1,2,4-oxadiazoles in the discovery of 1H-indazole-bearing neuroprotective MAO B inhibitors
Articolo
Carbohydrate-naphthalene diimide conjugates as potential antiparasitic drugs: Synthesis, evaluation and structure-activity studies
Articolo
Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents.
Articolo
Chemoenzymatically synthesized ganglioside GM3 analogues with inhibitory effects on tumor cell growth and migration
Articolo
Cholinergic agents structurally related to furtrethonium I
Articolo
Combining BNCT with carbonic anhydrase inhibition for mesothelioma treatment: Synthesis, in vitro, in vivo studies of ureidosulfamido carboranes
Articolo
Cyclic and branched acyl chain galactoglycerolipids and their effect on anti-tumor-promoting activity
Articolo
Design and synthesis of novel chalcones as potent selective monoamine oxidase-B inhibitors.
Articolo
Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis.
Articolo
Design, synthesis and biological evaluation of biphenylamide derivatives as Hsp90 C-terminal inhibitors
Articolo
Design, synthesis and evaluation of covalent inhibitors of DprE1 as antitubercular agents
Articolo
Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth.
Articolo
Development of QSAR models for predicting hepatocarcinogenic toxicity of chemicals
Articolo
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells
Articolo
Discovery and development of novel salicylate synthase (MbtI) furanic inhibitors as antitubercular agents
Articolo
Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics
Articolo
Discovery of new potent dual sigma receptor/GluN2b ligands with antioxidant property as neuroprotective agents
Articolo
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer
Articolo
Fibrate-derived N-(methylsulfonyl)amides with antagonistic properties on PPARa
Articolo
Glycoglycerolipid analogues active as anti-tumor-promoters: the influence of the anomeric configuration
Articolo
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign
Articolo
Identification of dual Sigma1 receptor modulators/acetylcholinesterase inhibitors with antioxidant and neurotrophic properties, as neuroprotective agents
Articolo
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group
Articolo
Merging memantine and ferulic acid to probe connections between NMDA receptors, oxidative stress and amyloid-β peptide in Alzheimer's disease
Articolo
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds
Articolo
Natural products against key Mycobacterium tuberculosis enzymatic targets: Emerging opportunities for drug discovery
Articolo
Novel S1R agonists counteracting NMDA excitotoxicity and oxidative stress: A step forward in the discovery of neuroprotective agents
Articolo
Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models
Articolo
Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis.
Articolo
Pyrrolo[3′,2′:6,7]cyclohepta[1,2-b]pyridines with potent photo-antiproliferative activity
Articolo
Rational design of allosteric modulators of the aromatase enzyme: An unprecedented therapeutic strategy to fight breast cancer
Articolo
Structural development studies of PPARs ligands based on tyrosine scaffold
Articolo
Substituted benzo[d]oxazol-2(3H)-one derivatives with preference for the sigma1 binding site
Articolo
Substituted benzylaminoalkylindoles with preference for the sigma2 binding site
Articolo
Synthesis and antiproliferative mechanism of action of pyrrolo[3′,2′:6,7] cyclohepta[1,2-d]pyrimidin-2-amines as singlet oxygen photosensitizers
Articolo
Synthesis and biological activities of triazole derivatives as inhibitors of InhA and antituberculosis agents
Articolo
Synthesis and biological evaluation of new aryl-alkyl(alkenyl)-4-benzylpiperidines, novel Sigma Receptor (SR) modulators, as potential anticancer-agents
Articolo
Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazoles as inhibitors of Mycobacterium tuberculosis
Articolo
Synthesis and photocytotoxic activity of [1,2,3]triazolo[4,5-h][1,6]naphthyridines and [1,3]oxazolo[5,4-h][1,6]naphthyridines
Articolo
Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis
Articolo
Synthesis, biological activity and mechanistic insights of 1-substituted cyclopropylamine derivatives: a novel class of irreversible inhibitors of histone demethylase KDM1A.
Articolo
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold
Articolo
The cell division protein FtsZ as a cellular target to hit cystic fibrosis pathogens
Articolo
The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents
Articolo
The opioid-receptor-like 1 (ORL-1) as a potential target for new analgesics
Articolo
Thiosugar naphthalene diimide conjugates: G-quadruplex ligands with antiparasitic and anticancer activity
Articolo
Virtual screening and crystallographic studies reveal an unexpected γ-lactone derivative active against MptpB as a potential antitubercular agent
Articolo
No Results Found
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